TargetMol

CAY10471 Racemate

Product Code:
 
TAR-T7359
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T7359-1mg1mg£95.00
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TAR-T7359-2mg2mg£106.00
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TAR-T7359-5mg5mg£128.00
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TAR-T7359-1mL1 mL * 10 mM (in DMSO)£134.00
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TAR-T7359-10mg10mg£161.00
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TAR-T7359-25mg25mg£262.00
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TAR-T7359-50mg50mg£356.00
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TAR-T7359-100mg100mg£494.00
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Further Information

Bioactivity:
CAY 10471 is a potent, highly selective CRTH2/DP 2 receptor antagonist. CAY10471 binds to the human CRTH2/DP2, DP1, and TP receptors( Ki values of 0.6, 1200, and >10,000 nM,respectively)
CAS:
844639-57-2
Formula:
C21H21FN2O4S
Molecular Weight:
416.47
Pathway:
Endocrinology/Hormones; Immunology/Inflammation; GPCR/G Protein
Purity:
0.98
SMILES:
CN(C1CCc2c(C1)c1ccccc1n2CC(O)=O)S(=O)(=O)c1ccc(F)cc1
Target:
GPR; Prostaglandin Receptor

References

Ulven T , Kostenis E . Minor Structural Modifications Convert the Dual TP/CRTH2 Antagonist Ramatroban into a Highly Selective and Potent CRTH2 Antagonist[J]. Journal of Medicinal Chemistry, 2005, 48(4):897-900.