TargetMol

KG-501

Product Code:
 
TAR-T7297
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
❮❯

No additional charges, what you see is what you pay! *

CodeSizePrice
TAR-T7297-2mg2mg£95.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T7297-5mg5mg£107.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T7297-1mL1 mL * 10 mM (in DMSO)£111.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T7297-10mg10mg£122.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T7297-50mg50mg£187.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T7297-100mg100mg£243.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
Prices exclude any Taxes / VAT
How to order with us   Contact us
Stay in control of your spending. These prices have no additional charges, not even shipping!
* Rare exceptions are clearly labelled (only 0.14% of items!).
Multibuy discounts available! Contact us to find what you can save.
This product comes from: United States.
Typical lead time: 10-14 working days.
Contact us for more accurate information.
  • Further Information
  • Documents
  • References
  • Show All

Further Information

Bioactivity:
KG-501 is a cAMP response element-binding protein (CREB) inhibitor(IC50 : 6.89 μM).
CAS:
18228-17-6
Formula:
C17H13ClNO5P
Molecular Weight:
377.72
Pathway:
Chromatin/Epigenetic
Purity:
0.98
SMILES:
OP(O)(=O)Oc1cc2ccccc2cc1C(=O)Nc1ccc(Cl)cc1
Target:
Epigenetic Reader Domain

References

Best J L , Amezcua C A , Mayr B , et al. Identification of small-molecule antagonists that inhibit an activator:coactivator interaction[J]. Proceedings of the National Academy of Sciences, 2004, 101(51):17622-17627. Kaori K , Haruka F , Hitomi S , et al. The Traditional Japanese Herbal Medicine Hachimijiogan Elicits Neurite Outgrowth Effects in PC12 Cells and Improves Cognitive in AD Model Rats via Phosphorylation of CREB[J]. Frontiers in Pharmacology, 2017, 8:850-.