TargetMol

LJI308

Product Code:
 
TAR-T6878
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T6878-1mg1mg£101.00
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TAR-T6878-5mg5mg£136.00
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TAR-T6878-1mL1 mL * 10 mM (in DMSO)£142.00
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TAR-T6878-10mg10mg£149.00
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TAR-T6878-25mg25mg£251.00
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TAR-T6878-50mg50mg£352.00
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Quantity:
TAR-T6878-100mg100mg£504.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
LJI308 is a potent, and pan-RSK (p90 ribosomal S6 kinase) inhibitor with IC50 of 6 nM, 4 nM, and 13 nM for RSK1, RSK2, and RSK3, respectively.
CAS:
1627709-94-7
Formula:
C21H18F2N2O2
Molecular Weight:
368.384
Pathway:
MAPK; PI3K/Akt/mTOR signaling
Purity:
0.9886
SMILES:
Oc1c(F)cc(cc1F)-c1cnccc1-c1ccc(cc1)N1CCOCC1
Target:
S6 Kinase

References

Aronchik I, et al. Mol Cancer Res. 2014, 12(5), 803-812. Davies AH, et al. Oncotarget. 2015, 6(24), 20570-205777.