TargetMol

AZ6102

Product Code:
 
TAR-T6768
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T6768-2mg2mg£100.00
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TAR-T6768-5mg5mg£118.00
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TAR-T6768-1mL1 mL * 10 mM (in DMSO)£124.00
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TAR-T6768-10mg10mg£148.00
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TAR-T6768-25mg25mg£256.00
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TAR-T6768-50mg50mg£367.00
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Quantity:
TAR-T6768-100mg100mg£511.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
AZ6102 is a potent TNKS1/2 inhibitor that has 100-fold selectivity against other PARP family enzymes and shows IC50 of 5 nM for Wnt pathway inhibition in DLD-1 cells.
CAS:
1645286-75-4
Formula:
C25H28N6O
Molecular Weight:
428.54
Pathway:
DNA Damage/DNA Repair; Chromatin/Epigenetic; Stem Cells; Cytoskeletal Signaling
Purity:
0.9991
SMILES:
C[C@H]1CN(C[C@@H](C)N1)c1cc(C)c(cn1)-c1ccc(cc1)-c1nc2n(C)ccc2c(=O)[nH]1
Target:
PARP; Wnt/beta-catenin

References

de Vicente J. et al. ACS Med Chem Lett. 2015, 6(9):1019-1024. Johannes JW,et al. ACS Med Chem Lett. 2015, 6(3):254-259.