TargetMol

(R)-Nepicastat HCl

Product Code:
 
TAR-T6356
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T6356-1mL1 mL * 10 mM (in DMSO)£179.00
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TAR-T6356-5mg5mg£179.00
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TAR-T6356-10mg10mg£254.00
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TAR-T6356-25mg25mg£417.00
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TAR-T6356-50mg50mg£540.00
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TAR-T6356-100mg100mg£757.00
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Further Information

Bioactivity:
(R)-Nepicastat HCl, the R-enantiomer of Nepicastat HCl, is a potent and selective inhibitor with IC50 of 25.1 nM and 18.3 nM for bovine and human dopamine-β-hydroxylase, with negligible affinity for twelve other enzymes and thirteen neurotransmitter receptors.
CAS:
195881-94-8
Formula:
C14H16ClF2N3S
Molecular Weight:
331.81
Pathway:
Metabolism
Purity:
0.98
SMILES:
Cl.NCc1c[nH]c(=S)n1[C@@H]1CCc2c(F)cc(F)cc2C1
Target:
Hydroxylase

References

Stanley WC, et al. Br J Pharmacol. 1997, 121(8), 1803-1809.