TargetMol

Birabresib

Product Code:
 
TAR-T6032
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T6032-2mg2mg£103.00
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TAR-T6032-5mg5mg£124.00
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TAR-T6032-1mL1 mL * 10 mM (in DMSO)£128.00
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TAR-T6032-10mg10mg£140.00
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TAR-T6032-25mg25mg£193.00
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TAR-T6032-50mg50mg£269.00
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TAR-T6032-100mg100mg£405.00
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TAR-T6032-200mg200mg£570.00
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TAR-T6032-500mg500mg£867.00
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This product comes from: United States.
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Further Information

Bioactivity:
Birabresib is a synthetic, small molecule inhibitor of the BET (Bromodomain and Extra-Terminal) family of bromodomain-containing proteins 2, 3 and 4 with potential antineoplastic activity.
CAS:
202590-98-5
Formula:
C25H22ClN5O2S
Molecular Weight:
491.99
Pathway:
Chromatin/Epigenetic
Purity:
0.9993
SMILES:
Cc1sc-2c(c1C)C(=N[C@@H](CC(=O)Nc1ccc(O)cc1)c1nnc(C)n-21)c1ccc(Cl)cc1
Target:
Epigenetic Reader Domain

References

Zhang G M, Huang S S, Ye L X, et al. Reciprocal positive regulation between BRD4 and YAP in GNAQ-mutant uveal melanoma cells confers sensitivity to BET inhibitors. Pharmacological Research. 2022: 106464. Boi M, et al. Mol Cancer Ther. 2013, 12, A219. Noel JK, et al. Mol Cancer Ther. 2013, 12, C244.