TargetMol

Elagolix sodium

Product Code:
 
TAR-T5031
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T5031-2mg2mg£101.00
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TAR-T5031-5mg5mg£119.00
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TAR-T5031-1mL1 mL * 10 mM (in DMSO)£142.00
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TAR-T5031-10mg10mg£148.00
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TAR-T5031-25mg25mg£211.00
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TAR-T5031-50mg50mg£301.00
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TAR-T5031-100mg100mg£430.00
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Further Information

Bioactivity:
Elagolix sodium is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).
CAS:
832720-36-2
Formula:
C32H29F5N3NaO5
Molecular Weight:
653.582
Pathway:
GPCR/G Protein
Purity:
0.9993
SMILES:
[Na+].COc1cccc(c1F)-c1c(C)n(Cc2c(F)cccc2C(F)(F)F)c(=O)n(CC(NCCCC([O-])=O)c2ccccc2)c1=O
Target:
GNRH Receptor

References

Barra F, Scala C, Ferrero S2.Elagolix sodium for the treatment of women with moderate to severe endometriosis-associated pain.Drugs Today (Barc). 2019 Apr;55(4):237-246. Elagolix (Orilissa)--an oral GnRH antagonist for endometriosis pain.[J]. The Medical letter on drugs and therapeutics, 2018.