TargetMol

Mequitazine

Product Code:
 
TAR-T4499
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T4499-5mg5mg£104.00
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TAR-T4499-1mL1 mL * 10 mM (in DMSO)£107.00
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TAR-T4499-10mg10mg£117.00
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TAR-T4499-25mg25mg£144.00
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TAR-T4499-50mg50mg£170.00
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TAR-T4499-100mg100mg£196.00
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Further Information

Bioactivity:
Mequitazine is an effective, nonsedative and long-acting histamine H1 antagonist.
CAS:
29216-28-2
Formula:
C20H22N2S
Molecular Weight:
322.47
Pathway:
Immunology/Inflammation; GPCR/G Protein; Neuroscience
Purity:
0.9995
SMILES:
C(C1CN2CCC1CC2)N1c2ccccc2Sc2ccccc12
Target:
Histamine Receptor

References

Gonnot V, et al. Expedient synthesis of mequitazine an antihistaminic drug by palladium catalyzed allylic alkylation of sodium phenothiazinate. Chem Pharm Bull (Tokyo). 2009 Nov;57(11):1300-2. Martinez-Mir I, et al. Antihistaminic and anticholinergic activities of mequitazine in comparison with clemizole. J Pharm Pharmacol. 1988 Sep;40(9):655-6. Satake N, et al. Possible mechanisms of vasoinhibitory effects of mequitazine, an antiallergic agent, on the contractions of isolated rat aorta induced by K+, phenylephrine, 5-hydroxytryptamine, and Ca2+. J Cardiovasc Pharmacol. 1994 Apr;23(4):669-73. El-Nakeeb MA, et a. In vitro antibacterial activity of some antihistaminics belonging to different groups against multi-drug resistant clinical isolates. Braz J Microbiol. 2011 Jul;42(3):980-91.