TargetMol

EPZ020411 2HCl (1700663-41-7(free base))

Product Code:
 
TAR-T4334
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T4334-2mg2mg£157.00
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TAR-T4334-5mg5mg£225.00
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TAR-T4334-1mL1 mL * 10 mM (in DMSO)£316.00
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TAR-T4334-10mg10mg£316.00
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TAR-T4334-25mg25mg£584.00
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This product comes from: United States.
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Further Information

Bioactivity:
EPZ020411 is an effective and specific small molecule PRMT6 inhibitor (IC50=10 nM).
CAS:
T4334
Formula:
C25H40Cl2N4O3
Molecular Weight:
515.51
Pathway:
Chromatin/Epigenetic
Purity:
0.992
SMILES:
Cl.Cl.CNCCN(C)Cc1c[nH]nc1-c1ccc(O[C@H]2C[C@@H](C2)OCCC2CCOCC2)cc1
Target:
Histone Methyltransferase

References

Mitchell LH, et al. Aryl Pyrazoles as Potent Inhibitors of Arginine Methyltransferases: Identification of the First PRMT6 ToolCompound. ACS Med Chem Lett. 2015 Apr 6;6(6):655-659.