TargetMol

PKM2-IN-1

Product Code:
 
TAR-T4170
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T4170-1mg1mg£98.00
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TAR-T4170-2mg2mg£108.00
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TAR-T4170-5mg5mg£132.00
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TAR-T4170-1mL1 mL * 10 mM (in DMSO)£139.00
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TAR-T4170-10mg10mg£164.00
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TAR-T4170-25mg25mg£244.00
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TAR-T4170-50mg50mg£369.00
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TAR-T4170-100mg100mg£550.00
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Quantity:
TAR-T4170-200mg200mg£755.00
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Quantity:
TAR-T4170-500mg500mg£1,107.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
PKM2 inhibitor(Compound 3K) displays PKM2 inhibitory activity with the IC50 value of 2.95 μM. The IC50 value for PKM1 is 4-5-fold higher than that for PKM2.
CAS:
94164-88-2
Formula:
C18H19NO2S2
Molecular Weight:
345.48
Pathway:
Metabolism
Purity:
0.999
SMILES:
CC1=C(CSC(=S)N2CCCCC2)C(=O)c2ccccc2C1=O
Target:
PKM

References

Ning X, et al. Discovery of novel naphthoquinone derivatives as inhibitors of the tumor cell specific M2 isoform of pyruvate kinase. Eur J Med Chem. 2017 Sep 29;138:343-352.