TargetMol

XMD8-87

Product Code:
 
TAR-T3709
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T3709-2mg2mg£102.00
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TAR-T3709-5mg5mg£128.00
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TAR-T3709-1mL1 mL * 10 mM (in DMSO)£134.00
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TAR-T3709-10mg10mg£172.00
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TAR-T3709-25mg25mg£298.00
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TAR-T3709-50mg50mg£436.00
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TAR-T3709-100mg100mg£610.00
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TAR-T3709-500mg500mg£1,219.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
XMD8-87 is a TNK2 inhibitor with activity in the inhibition of TNK2 phosphorylation. XMD8-87 and XMD16-5 potently inhibit phosphorylation of TNK2 truncation mutations found in solid tumor types.
CAS:
1234480-46-6
Formula:
C24H27N7O2
Molecular Weight:
445.527
Pathway:
DNA Damage/DNA Repair; Metabolism; Proteases/Proteasome
Purity:
0.9761
SMILES:
COc1cc(ccc1Nc1ncc2NC(=O)c3ccccc3N(C)c2n1)N1CCN(C)CC1
Target:
Tyrosinase; PPAR

References

Maxson JE, et al. Cancer Res. 2016, 76(1):127-38.