TargetMol

MK-4827 Racemate

Product Code:
 
TAR-T22988
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T22988-1mg1mg£107.00
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TAR-T22988-2mg2mg£121.00
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TAR-T22988-5mg5mg£142.00
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TAR-T22988-1mL1 mL * 10 mM (in DMSO)£168.00
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TAR-T22988-10mg10mg£196.00
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TAR-T22988-25mg25mg£309.00
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TAR-T22988-50mg50mg£487.00
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TAR-T22988-100mg100mg£631.00
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Further Information

Bioactivity:
MK-4827 Racemate is a selective PARP1 and PARP2 inhibitor with IC50s of 3.8 nM and 2.1 nM, respectively, over 330-fold selectivity for PARP3, V-PARP and Tank1.
CAS:
1038915-75-1
Formula:
C19H20N4O
Molecular Weight:
320.396
Pathway:
DNA Damage/DNA Repair; Chromatin/Epigenetic
Purity:
0.9947
SMILES:
NC(=O)c1cccc2cn(nc12)-c1ccc(cc1)C1CCCNC1
Target:
PARP

References

1. Sch?fer P, Palacin T, Sidera M, Fletcher SP. Asymmetric Suzuki-Miyaura coupling of heterocycles via Rhodium-catalysed allylic arylation of racemates. Nat Commun. 2017 Jun 13;8:15762.