TargetMol

CID 2745687

Product Code:
 
TAR-T21874
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T21874-1mg1mg£98.00
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Quantity:
TAR-T21874-2mg2mg£109.00
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TAR-T21874-5mg5mg£135.00
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Quantity:
TAR-T21874-1mL1 mL * 10 mM (in DMSO)£142.00
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Quantity:
TAR-T21874-10mg10mg£173.00
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Quantity:
TAR-T21874-25mg25mg£303.00
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Quantity:
TAR-T21874-50mg50mg£436.00
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Quantity:
TAR-T21874-100mg100mg£610.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
CID 2745687 is a GPR35 antagonist that inhibited the effects at human GPR35 of cromolyn disodium and zaprinast, two agonists that share an overlapping binding site.
CAS:
264233-05-8
Formula:
C17H19F2N5O2S
Molecular Weight:
395.43
Pathway:
GPCR/G Protein; Endocrinology/Hormones
Purity:
0.9911
SMILES:
COC(=O)c1cnn(c1C=NNC(=S)NC(C)(C)C)-c1ccc(F)cc1F
Target:
GPR

References

1. Jenkins L , Harries N , Lappin J E , et al. Antagonists of GPR35 display high species ortholog selectivity and varying modes of action[J]. Journal of Pharmacology & Experimental Therapeutics, 2012, 343(3):683-695.