TargetMol

N-desmethyl Enzalutamide

Product Code:
 
TAR-T19450
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T19450-1mg1mg£98.00
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TAR-T19450-2mg2mg£109.00
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TAR-T19450-5mg5mg£135.00
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TAR-T19450-1mL1 mL * 10 mM (in DMSO)£142.00
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TAR-T19450-10mg10mg£161.00
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TAR-T19450-25mg25mg£258.00
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TAR-T19450-50mg50mg£431.00
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TAR-T19450-100mg100mg£600.00
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TAR-T19450-500mg500mg£1,187.00
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This product comes from: United States.
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Further Information

Bioactivity:
N-desmethyl Enzalutamide is the active Enzalutamide metabolite.It is the active metabolite of Enzalutamide. N-desmethyl Enzalutamide demonstrates primary and secondary pharmacodynamics of similar potency to Enzalutamide and circulates at approximately the same plasma concentrations as enzalutamide.
CAS:
1242137-16-1
Formula:
C20H14F4N4O2S
Molecular Weight:
450.41
Pathway:
Endocrinology/Hormones
Purity:
0.9962
SMILES:
CC1(C)N(C(=S)N(C1=O)c1ccc(C#N)c(c1)C(F)(F)F)c1ccc(C(N)=O)c(F)c1
Target:
Androgen Receptor

References

1. Gibbons JA, et al. Pharmacokinetic Drug Interaction Studies with Enzalutamide. Clin Pharmacokinet. 2015 Oct;54(10):1057-69.