TargetMol

Thiethylperazine dimaleate

Product Code:
 
TAR-T17072
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T17072-1mg1mg£98.00
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TAR-T17072-5mg5mg£135.00
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TAR-T17072-10mg10mg£168.00
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TAR-T17072-25mg25mg£249.00
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TAR-T17072-50mg50mg£369.00
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TAR-T17072-100mg100mg£530.00
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Quantity:
TAR-T17072-500mg500mg£1,026.00
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This product comes from: United States.
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Further Information

Bioactivity:
Thiethylperazine dimaleate is an antagonist of the D2 receptor and H1 receptor. Thiethylperazine dimaleate is an activator of ABCC1 and possesses antimicrobial, anti-emetic, and antipsychotic effects.
CAS:
1179-69-7
Formula:
C30H37N3O8S2
Molecular Weight:
631.76
Pathway:
Neuroscience; Immunology/Inflammation; Membrane transporter/Ion channel; Microbiology/Virology; GPCR/G Protein
Purity:
0.98
SMILES:
OC(=O)C=C/C(O)=O.OC(=O)C=C/C(O)=O.CCSc1ccc2Sc3ccccc3N(CCCN3CCN(C)CC3)c2c1
Target:
Dopamine Receptor; Antibacterial; ABC; Histamine Receptor

References

1. Czeizel AE, et al. Case-control study of teratogenic potential of thiethylperazine, an anti-emetic drug. BJOG. 2003 May;110(5):497-9. 2. Krohn M, et al. Cerebral amyloid-? proteostasis is regulated by the membrane transport protein ABCC1 in mice. J Clin Invest. 2011 Oct;121(10):3924-31. 3. Rahbar M, et al. Enhancement of vancomycin activity by phenothiazines against vancomycin-resistant Enterococcus faecium in vitro. Basic Clin Pharmacol Toxicol. 2010 Aug;107(2):676-9.