TargetMol

PF-5190457

Product Code:
 
TAR-T16508
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T16508-50mg50mgEnquire
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TAR-T16508-1mg1mg£95.00
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TAR-T16508-2mg2mg£106.00
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TAR-T16508-5mg5mg£128.00
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TAR-T16508-1mL1 mL * 10 mM (in DMSO)£136.00
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TAR-T16508-10mg10mg£173.00
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TAR-T16508-25mg25mg£303.00
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Further Information

Bioactivity:
PF-5190457 is an effective and selective ghrelin receptor inverse agonist (pKi: 8.36).
CAS:
1334782-79-4
Formula:
C29H32N6OS
Molecular Weight:
512.68
Pathway:
GPCR/G Protein
Purity:
0.9934
SMILES:
Cc1cn2cc(CC(=O)N3CCC4(CN(C4)[C@@H]4CCc5cc(ccc45)-c4cc(C)ncn4)CC3)nc2s1
Target:
GHSR

References

1. Bhattacharya SK, et al. Discovery of PF-5190457, a Potent, Selective, and Orally Bioavailable Ghrelin Receptor Inverse Agonist Clinical Candidate. ACS Med Chem Lett. 2014 Feb 24;5(5):474-9.