TargetMol

CVT-10216

Product Code:
 
TAR-T15022
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T15022-1mg1mg£105.00
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TAR-T15022-5mg5mg£148.00
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TAR-T15022-1mL1 mL * 10 mM (in DMSO)£160.00
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TAR-T15022-10mg10mg£212.00
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TAR-T15022-25mg25mg£356.00
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TAR-T15022-50mg50mg£527.00
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Quantity:
TAR-T15022-100mg100mg£724.00
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Further Information

Bioactivity:
CVT-10216 is a Potent and selective, reversible inhibitor of aldehyde dehydrogenase 2 (ALDH2) (IC50: 29 nM). CVT-10216 also has inhibitory effect of ALDH-1 (IC50: 1.3 μM). CVT-10216 can reduce excessive alcohol drinking in alcohol-preferring rats and exhibit anxiolytic effects.
CAS:
1005334-57-5
Formula:
C24H19NO7S
Molecular Weight:
465.48
Pathway:
Metabolism
Purity:
0.9916
SMILES:
CS(=O)(=O)Nc1ccc(cc1)-c1coc2cc(OCc3cccc(c3)C(O)=O)ccc2c1=O
Target:
Dehydrogenase

References

1. Overstreet DH, et al. A selective ALDH-2 inhibitor reduces anxiety in rats.Pharmacol Biochem Behav. 2009 Dec;94(2):255-61.