TargetMol

CCG-63808

Product Code:
 
TAR-T14898
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T14898-25mg25mgEnquire
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TAR-T14898-50mg50mgEnquire
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TAR-T14898-1mg1mg£105.00
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TAR-T14898-2mg2mg£120.00
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TAR-T14898-5mg5mg£148.00
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TAR-T14898-10mg10mg£201.00
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Further Information

Bioactivity:
CCG-63808 is a reversible inhibitor of regulator of G-protein signaling (RGS) proteins. CCG-63808 dose-dependently inhibits the TR-FRET signal between RGS4-AF488 and Tb-Gαo with IC50 values of 1.9 μM.
CAS:
620113-73-7
Formula:
C25H15FN4O2S
Molecular Weight:
454.48
Pathway:
GPCR/G Protein
Purity:
0.98
SMILES:
Cc1cccn2c1nc(Oc1ccc(F)cc1)c(C=C(/C#N)c1nc3ccccc3s1)c2=O
Target:
GTPase

References

1. Levi L. Blazer et al.Reversible, Allosteric Small-Molecule Inhibitors of Regulator of G Protein Signaling Proteins. Molecular Pharmacology September 2010 vol.78 no.3 524-533