TargetMol

AKR1C1-IN-1

Product Code:
 
TAR-T14151
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T14151-1mg1mg£106.00
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TAR-T14151-2mg2mg£122.00
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TAR-T14151-5mg5mg£149.00
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TAR-T14151-1mL1 mL * 10 mM (in DMSO)£164.00
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TAR-T14151-10mg10mg£201.00
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TAR-T14151-25mg25mg£306.00
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TAR-T14151-50mg50mg£454.00
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TAR-T14151-100mg100mg£623.00
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Quantity:
TAR-T14151-500mg500mg£1,211.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
AKR1C1-IN-1 is a human 20α-hydroxysteroid dehydrogenase (AKR1C1) inhibitor (Ki: 4 nM for AKR1C1).
CAS:
4906-68-7
Formula:
C13H9BrO3
Molecular Weight:
293.116
Pathway:
Metabolism
Purity:
0.9946
SMILES:
OC(=O)c1cc(cc(Br)c1O)-c1ccccc1
Target:
NADPH

References

1. El-Kabbani O, et al. Structure-guided design, synthesis, and evaluation of salicylic acid-based inhibitors targeting a selectivity pocket in the active site of human 20alpha-hydroxysteroid dehydrogenase (AKR1C1). J Med Chem. 2009 May 28;52(10):3259-64.