TargetMol

PKC-IN-1

Product Code:
 
TAR-T12494
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T12494-5mg5mg£351.00
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Quantity:
TAR-T12494-50mg50mg£1,267.00
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Quantity:
TAR-T12494-100mg100mg£1,669.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
PKC-IN-1 is an ATP-competitive and reversible conventional PKC enzymes inhibitor (PKCα, PKCβI, PKCβII, PKC?, PKCγ, PKC mu and PKCε with IC50s of 2.3, 8.1, 7.6, 25.6, 57.5, 314, 808 nM, respectively).
CAS:
1046787-18-1
Formula:
C25H37FN8O2
Molecular Weight:
500.623
Pathway:
Cytoskeletal Signaling; Chromatin/Epigenetic
Purity:
0.98
SMILES:
C[C@@H]1CN([C@@H](C)CN1CC1CCOCC1)C(=O)N1Cc2c(Nc3nc(C)ncc3F)n[nH]c2C1(C)C
Target:
PKC

References

1. Michael Niesman, et al. Treatment of autoimmune disease. WO2015179847A1.