TargetMol

EPZ031686

Product Code:
 
TAR-TQ0263
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
❮❯

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CodeSizePrice
TAR-TQ0263-1mg1mg£189.00
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TAR-TQ0263-2mg2mg£242.00
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TAR-TQ0263-5mg5mg£349.00
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TAR-TQ0263-1mL1 mL * 10 mM (in DMSO)£434.00
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TAR-TQ0263-10mg10mg£470.00
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TAR-TQ0263-25mg25mg£707.00
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TAR-TQ0263-50mg50mg£978.00
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TAR-TQ0263-100mg100mg£1,291.00
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Further Information

Bioactivity:
EPZ031686 is an effective inhibitor of SMYD3 inhibitor with an IC50 of 3 nM and can be used in studies about cancer.
CAS:
1808011-22-4
Formula:
C26H34ClF3N4O4S
Molecular Weight:
591.09
Pathway:
Chromatin/Epigenetic
Purity:
0.9791
SMILES:
[H][C@]12CC[C@]([H])(C[C@@]([H])(C1)NC(=O)c1cc3CC(=O)Nc3cc1Cl)N2S(=O)(=O)CC1CCN(CCCC(F)(F)F)CC1
Target:
Histone Methyltransferase

References

Mitchell LH et al. Novel Oxindole Sulfonamides and Sulfamides: EPZ031686, the First Orally Bioavailable Small Molecule SMYD3 Inhibitor. ACS Med Chem Lett. 2015 Aug 27;7(2):134-8.