TargetMol

UFP-101 acetate

Product Code:
 
TAR-TP2105L
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-TP2105L-1mg1mg£325.00
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TAR-TP2105L-2mg2mg£531.00
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TAR-TP2105L-5mg5mg£791.00
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TAR-TP2105L-10mg10mg£1,058.00
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TAR-TP2105L-25mg25mg£1,532.00
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TAR-TP2105L-50mg50mg£2,046.00
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Quantity:
TAR-TP2105L-100mg100mg£2,713.00
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This product comes from: United States.
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Further Information

Bioactivity:
UFP-101 acetate is a selective and competitive antagonist of the NOP receptor (pKi = 10.24) with >3000-fold selectivity over δ, μ, and κ opioid receptors.
CAS:
TP2105L
Formula:
C84H142N32O23
Molecular Weight:
1968.23
Pathway:
GPCR/G Protein; Neuroscience; Endocrinology/Hormones
Purity:
0.9592
SMILES:
CC(O)=O.O=C(N)[C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC(CNC([C@@H](NC([C@@H](NC(CNC(CNC(CNCC1=CC=CC=C1)=O)=O)=O)CC2=CC=CC=C2)=O)[C@H](O)C)=O)=O)C)=O)CCCNC(N)=N)=O)CCCCN)=O)CO)=O)C)=O)CCCNC(N)=N)=O)CCCCN)=O)CCCNC(N)=N)=O)CCCCN)=O)CC(N)=O)=O)CCC(N)=O
Target:
Opioid Receptor

References

Gavioli EC, et al. Blockade of nociceptin/orphanin FQ-NOP receptor signalling produces antidepressant-like effects: pharmacological and genetic evidences from the mouse forced swimming test. Eur J Neurosci. 2003;17(9):1987-1990. Calo G, et al. [Nphe1,Arg14,Lys15]nociceptin-NH2, a novel potent and selective antagonist of the nociceptin/orphanin FQ receptor. Br J Pharmacol. 2002;136(2):303-311.