TargetMol

CTAP(TFA? (103429-32-9 free base)

Product Code:
 
TAR-TP2050L
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-TP2050L-1mg1mg£235.00
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TAR-TP2050L-5mg5mg£483.00
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TAR-TP2050L-10mg10mg£667.00
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TAR-TP2050L-25mg25mg£994.00
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TAR-TP2050L-50mg50mg£1,315.00
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Quantity:
TAR-TP2050L-100mg100mg£1,741.00
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Quantity:
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This product comes from: United States.
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Further Information

Bioactivity:
CTAP TFA is a potent, highly selective, and brain penetrant antagonist of μ-opioid receptor with IC50 of 3.5 nM. It displays over 1200-fold selectivity over δ opioid (IC50=4500 nM) and somatostatin receptors. CTAP TFA can be used for the study of L-DOPA-induced dyskinesia (LID)
CAS:
TP2050L
Formula:
C53H70F3N13O13S2
Molecular Weight:
1218.33
Pathway:
Endocrinology/Hormones; GPCR/G Protein; Neuroscience
Purity:
0.9962
SMILES:
CC(O)C1C(NC(C(NC(C(N)=O)C(O)C)=O)C(C)(C)SSCC(NC(C(N)CC2=CC=CC=C2)=O)C(NC(CC3=CC=C(O)C=C3)C(NC(CC4=CNC5=CC=CC=C54)C(NC(CCC/N=C(N)N)C(N1)=O)=O)=O)=O)=O.O=C(O)C(F)(F)F
Target:
Opioid Receptor

References

Mitchell J Bartlett, et al. Highly-selective ?-opioid Receptor Antagonism Does Not Block L-DOPA-induced Dyskinesia in a Rodent Model.BMC Res Notes