TargetMol

[Ala17]-MCH acetate

Product Code:
 
TAR-TP1997L
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-TP1997L-1mg1mg£229.00
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TAR-TP1997L-5mg5mg£463.00
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TAR-TP1997L-10mg10mg£643.00
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TAR-TP1997L-25mg25mg£946.00
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TAR-TP1997L-50mg50mg£1,259.00
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TAR-TP1997L-100mg100mg£1,661.00
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Quantity:
TAR-TP1997L-500mg500mg£3,259.00
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Further Information

Bioactivity:
[Ala17]-MCH acetate is a selective ligand for MCHR1 with a Ki of 0.16 nM and Kd of 0.37 nM(Eu3+ chelate-labeled). [Ala17]-MCH acetate shows selectivity over MCHR2 with Ki of 34 nM.
CAS:
TP1997L
Formula:
C99H159N29O28S4
Molecular Weight:
2331.76
Pathway:
GPCR/G Protein
Purity:
0.9892
SMILES:
O=C1N2[C@](CCC2)([H])C(N[C@@H](CSSC[C@@H](C(N[C@H](C(N[C@H](C(NCC(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H]1CCCNC(N)=N)=O)CC3=CC=C(C=C3)O)=O)C(C)C)=O)CCCNC(N)=N)=O)=O)CC(C)C)=O)CCSC)=O)NC([C@H](CCCNC(N)=N)NC([C@H](CC(C)C)NC([C@H](CCSC)NC([C@H](CC(O)=O)NC([C@@H](NC([C@@H](N)CC(O)=O)=O)CC4=CC=CC=C4)=O)=O)=O)=O)=O)C(N[C@@H](C)C(N[C@@H](CCC(N)=O)C(N[C@H](C(O)=O)C(C)C)=O)=O)=O)=O.CC(O)=O
Target:
Melanin-concentrating Hormone Receptor (MCHR)

References

Xiaoying Gao, et al. Europium-labeled melanin-concentrating hormone analogues: ligands for measuring binding to melanin-concentrating hormone receptors 1 and 2. Anal Biochem. 2004 May 15;328(2):187-95.