TargetMol

Ziconotide Acetate (107452-89-1 free base)

Product Code:
 
TAR-TP1559L
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
 

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CodeSizePrice
TAR-TP1559L-50mg50mgEnquire
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TAR-TP1559L-1mg1mg£211.00
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TAR-TP1559L-5mg5mg£369.00
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TAR-TP1559L-10mg10mg£503.00
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TAR-TP1559L-25mg25mg£759.00
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This product comes from: United States.
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Further Information

Bioactivity:
Ziconotide is an analgesic agent and has been used to treat neuropathic and non-neuropathic pain. Ziconotide acts by binding to N-type calcium channels situated on the terminal part of primary afferent neurons of the nociceptive pathway therefore reducing synaptic transmission with potent antinociceptive effects.
CAS:
914454-03-8
Formula:
C102H172N36O32S7
Molecular Weight:
2639.2
Pathway:
Metabolism; Membrane transporter/Ion channel
Purity:
0.9952
SMILES:
CC1C(=O)NC(C(=O)NC2CSSCC3C(=O)NC(C(=O)NC(C(=O)NCC(=O)NC(C(=O)NC(CSSCC(C(=O)NC(CSSCC(C(=O)NC(C(=O)NCC(=O)NC(C(=O)NCC(=O)N1)CCCCN)CCCCN)N)C(=O)NC(C(=O)NCC(=O)NC(C(=O)N3)CO)C(C)O)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC2=O)CO)CCCNC(=N)N)CC(C)C)CCSC
Target:
Calcium Channel

References

Brinzeu A, Berthiller J, Caillet JB, Staquet H, Mertens P. Ziconotide for spinal cord injury-related pain. Eur J Pain. 2019;23(9):1688-1700. doi:10.1002/ejp.1445 Dong Y, Gao Y, Xu S, et al. Closed-state inactivation and pore-blocker modulation mechanisms of human CaV2. 2. Cell Reports. 2021, 37(5): 109931.