TargetMol

FC131 TFA (606968-52-9 free base)

Product Code:
 
TAR-TP1348
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
❮❯

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CodeSizePrice
TAR-TP1348-1mg1mg£132.00
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TAR-TP1348-2mg2mg£179.00
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TAR-TP1348-5mg5mg£303.00
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TAR-TP1348-10mg10mg£460.00
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TAR-TP1348-25mg25mg£709.00
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TAR-TP1348-50mg50mg£978.00
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Quantity:
TAR-TP1348-100mg100mg£1,340.00
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Quantity:
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Further Information

Bioactivity:
FC131 TFA is an antagonist of CXCR4 that inhibits the binding of [125I] -sdf-1 to CXCR4(IC50 : 4.5 nM ), and has anti-hiv activity.
CAS:
TP1348
Formula:
C38H48F3N11O8
Molecular Weight:
843.85
Pathway:
Microbiology/Virology; Proteases/Proteasome; Autophagy; Immunology/Inflammation; GPCR/G Protein
Purity:
0.9967
SMILES:
FC(F)(F)C(=O)O.N=C(N)NCCC[C@@H]4NC(=O)[C@@H](NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](Cc2cc3ccccc3cc2)NC4=O)CCCNC(=N)N
Target:
HIV Protease; CXCR

References

Tamamura H, et al. Stereoselective synthesis of [L-Arg-L/D-3-(2-naphthyl)alanine]-type (E)-alkene dipeptide isosteres and its application to the synthesis and biological evaluation of pseudopeptide analogues of the CXCR4 antagonist FC131. J Med Chem. 2005 Jan 27;48(2):380-91.