TargetMol

CYN 154806 TFA(183658-72-2 free base)

Product Code:
 
TAR-TP1346
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
❮❯

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CodeSizePrice
TAR-TP1346-1mg1mg£189.00
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TAR-TP1346-5mg5mg£454.00
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TAR-TP1346-10mg10mg£624.00
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TAR-TP1346-25mg25mg£938.00
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TAR-TP1346-50mg50mg£1,259.00
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TAR-TP1346-100mg100mg£1,645.00
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Further Information

Bioactivity:
CYN 154806 TFA is a cyclic octapeptide and an effective selective somatostatin sst2 receptor antagonist. For the recombinant sst2, sst1, sst3, sst4 and sst5 receptors, the pIC50 values are 8.58, 5.41, 6.07, 5.76 and 6.48, respectively.
CAS:
TP1346
Formula:
C58H69F3N12O16S2
Molecular Weight:
1311.36
Pathway:
GPCR/G Protein
Purity:
0.997
SMILES:
C[C@@H](O)[C@H]1C(N[C@H](C(N[C@@H](C(N)=O)CC2=CC=C(O)C=C2)=O)CSSC[C@@H](NC([C@@H](NC(C)=O)CC3=CC=C([N+]([O-])=O)C=C3)=O)C(N[C@@H](CC4=CC=C(O)C=C4)C(N[C@H](CC5=CNC6=CC=CC=C65)C(N[C@@H](CCCCN)C(N1)=O)=O)=O)=O)=O.OC(C(F)(F)F)=O
Target:
Somatostatin

References

Bass RT, et al. Identification and characterization of novel somatostatin antagonists. Mol Pharmacol. 1996 Oct;50(4):709-15.