TargetMol

[Pyr1]-Apelin-13

Product Code:
 
TAR-TP1260
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-TP1260-1mg1mg£142.00
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TAR-TP1260-5mg5mg£303.00
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TAR-TP1260-10mg10mg£436.00
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TAR-TP1260-25mg25mg£662.00
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TAR-TP1260-50mg50mg£863.00
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Quantity:
TAR-TP1260-100mg100mg£1,163.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
[Pyr1]-Apelin-13 is a potent and selective endogenous Apelin receptor (APJ) agonist.
CAS:
217082-60-5
Formula:
C69H108N22O16S
Molecular Weight:
1533.82
Pathway:
GPCR/G Protein
Purity:
1
SMILES:
CSCCC(NC(=O)C1CCCN1C(=O)CNC(=O)C(CCCCN)NC(=O)C(Cc1c[nH]cn1)NC(=O)C(CO)NC(=O)C(CC(C)C)NC(=O)C(CCCNC(N)=N)NC(=O)C1CCCN1C(=O)C(CCCNC(N)=N)NC(=O)C1CCC(=O)N1)C(=O)N1CCCC1C(=O)NC(Cc1ccccc1)C(O)=O
Target:
Apelin receptor

References

Serpooshan V, et al. [Pyr1]-Apelin-13 delivery via nano-liposomal encapsulation attenuates pressure overload-induced cardiac dysfunction. Biomaterials. 2015 Jan;37:289-98. Song K, Yang X, An G, et al.Targeting APLN/APJ restores blood-testis barrier and improves spermatogenesis in murine and human diabetic models.Nature Communications.2022, 13(1): 1-17.