TargetMol

GSK199

Product Code:
 
TAR-T8861
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T8861-1mg1mg£310.00
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TAR-T8861-2mg2mg£389.00
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TAR-T8861-5mg5mg£540.00
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TAR-T8861-1mL1 mL * 10 mM (in DMSO)£662.00
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TAR-T8861-10mg10mg£742.00
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TAR-T8861-25mg25mg£1,091.00
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Quantity:
TAR-T8861-50mg50mg£1,452.00
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Quantity:
TAR-T8861-100mg100mg£1,910.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
GSK199 is a selective PAD4 inhibitor(IC50 of 200 nM in the absence of calcium).
CAS:
1549811-53-1
Formula:
C24H29ClN6O2
Molecular Weight:
468.99
Pathway:
Chromatin/Epigenetic
Purity:
0.9809
SMILES:
Cl.CCn1c(cc2cccnc12)-c1nc2cc(cc(OC)c2n1C)C(=O)N1CCC[C@@H](N)C1
Target:
PAD

References

Willis V C , Banda N K , Cordova K N , et al. Protein arginine deiminase 4 inhibition is sufficient for the amelioration of collagen-induced arthritis[J]. Clinical & Experimental Immunology, 2017.