TargetMol

EST64454 hydrochloride

Product Code:
 
TAR-T8834
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T8834-1mg1mg£179.00
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TAR-T8834-2mg2mg£226.00
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TAR-T8834-5mg5mg£298.00
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TAR-T8834-1mL1 mL * 10 mM (in DMSO)£338.00
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TAR-T8834-10mg10mg£434.00
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TAR-T8834-25mg25mg£669.00
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TAR-T8834-50mg50mg£914.00
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TAR-T8834-100mg100mg£1,187.00
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Further Information

Bioactivity:
EST64454 is a highly soluble σ1 receptor antagonist (Ki : 22 nM),has the potential for Pain Management.
CAS:
1950569-11-5
Formula:
C18H23ClF2N4O2
Molecular Weight:
400.85
Pathway:
GPCR/G Protein
Purity:
0.9915
SMILES:
Cl.CC(=O)N1CCN(CCOCc2ccn(n2)-c2ccc(F)c(F)c2)CC1
Target:
Sigma receptor

References

Jos? Luis D?az, M?nica Garc?a, Torrens A , et al. EST64454: a Highly Soluble ? 1 Receptor Antagonist Clinical Candidate for Pain Management[J]. Journal of Medicinal Chemistry, 2020, 63(23):14979-14988.