TargetMol

Clobenpropit dihydrobromide

Product Code:
 
TAR-T8439
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T8439-1mg1mg£101.00
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TAR-T8439-5mg5mg£142.00
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TAR-T8439-1mL1 mL * 10 mM (in DMSO)£157.00
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TAR-T8439-10mg10mg£195.00
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TAR-T8439-25mg25mg£349.00
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TAR-T8439-50mg50mg£542.00
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TAR-T8439-100mg100mg£744.00
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Further Information

Bioactivity:
Clobenpropit dihydrobromide is a potent antagonist and inverse agonist of histamine H3R (histamine H3LR,pEC50 of 8.07)
CAS:
145231-35-2
Formula:
C14H19Br2ClN4S
Molecular Weight:
470.7
Pathway:
Apoptosis; Neuroscience; Immunology/Inflammation; GPCR/G Protein
Purity:
0.9948
SMILES:
Br.Br.Clc1ccc(CNC(=N)SCCCc2cnc[nH]2)cc1
Target:
Apoptosis; Histamine Receptor

References

Mena-Avila E, et al. Clobenpropit, a histamine H3 receptor antagonist/inverse agonist, inhibits [3H]-dopamine uptake by human neuroblastoma SH-SY5Y cells and rat brain synaptosomes. Pharmacol Rep. 2018 Feb;70(1):146-155. Esbenshade TA, et al. Two novel and selective nonimidazole histamine H3 receptor antagonists A-304121 and A-317920: I. In vitro pharmacological effects. J Pharmacol Exp Ther. 2003 Jun;305(3):887-96.