TargetMol

TFLLR-NH2 2TFA(197794-83-5(free base))

Product Code:
 
TAR-T7573L
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T7573L-1mg1mg£177.00
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TAR-T7573L-5mg5mg£484.00
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TAR-T7573L-1mL1 mL * 10 mM (in DMSO)£631.00
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TAR-T7573L-10mg10mg£667.00
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TAR-T7573L-25mg25mg£978.00
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TAR-T7573L-50mg50mg£1,299.00
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Quantity:
TAR-T7573L-100mg100mg£1,661.00
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Further Information

Bioactivity:
TFLLR-NH2(2TFA) is an agonist of PAR1 (EC50 :1.9 μM).
CAS:
T7573L
Formula:
C35H55F6N9O10
Molecular Weight:
875.87
Pathway:
GPCR/G Protein
Purity:
1
SMILES:
OC(C(F)(F)F)=O.CC(C[C@@H](C(N[C@H](C(N)=O)CCCNC(N)=N)=O)NC([C@@H](NC([C@@H](NC([C@H]([C@H](O)C)N)=O)Cc1ccccc1)=O)CC(C)C)=O)C.OC(C(F)(F)F)=O
Target:
Protease-activated Receptor

References

Kawabata A , Kuroda R , Kuroki N , et al. Characterization of the protease-activated receptor-1-mediated contraction and relaxation in the rat duodenal smooth muscle[J]. Life Sciences, 2000, 67(20):0-2530. Jia Y , Zhang S , Miao L , et al. Activation of platelet protease-activated receptor-1 induces epithelial-mesenchymal transition and chemotaxis of colon cancer cell line SW620[J]. Oncology Reports, 2015.