TargetMol

GSK1324726A

Product Code:
 
TAR-T6021
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T6021-1mg1mg£102.00
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TAR-T6021-2mg2mg£115.00
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TAR-T6021-5mg5mg£145.00
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TAR-T6021-1mL1 mL * 10 mM (in DMSO)£149.00
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TAR-T6021-10mg10mg£201.00
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TAR-T6021-25mg25mg£303.00
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TAR-T6021-50mg50mg£445.00
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TAR-T6021-100mg100mg£619.00
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TAR-T6021-500mg500mg£1,235.00
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Further Information

Bioactivity:
GSK1324726A is a greatly specific inhibitor of BET family proteins for BRD2(IC50=41 nM), BRD3(IC50=31 nM), and BRD4 (IC50=22 nM).
CAS:
1300031-52-0
Formula:
C25H23ClN2O3
Molecular Weight:
434.92
Pathway:
Apoptosis; Chromatin/Epigenetic
Purity:
0.9834
SMILES:
C[C@H]1C[C@@H](Nc2ccc(Cl)cc2)c2cc(ccc2N1C(C)=O)-c1ccc(cc1)C(O)=O
Target:
Apoptosis; Epigenetic Reader Domain

References

Gosmini R, et al. J Med Chem. 2014, 57(19), 8111-8131. Wyce A, et al. PLoS One. 2013, 8(8), e72967.