TargetMol

TAPI-1 trifluoroacetate (163847-77-6(free base))

Product Code:
 
TAR-T4122
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
❮❯

No additional charges, what you see is what you pay! *

CodeSizePrice
TAR-T4122-1mg1mg£189.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T4122-2mg2mg£285.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T4122-5mg5mg£546.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
Prices exclude any Taxes / VAT
How to order with us   Contact us
Stay in control of your spending. These prices have no additional charges, not even shipping!
* Rare exceptions are clearly labelled (only 0.14% of items!).
Multibuy discounts available! Contact us to find what you can save.
This product comes from: United States.
Typical lead time: 10-14 working days.
Contact us for more accurate information.
  • Further Information
  • Documents
  • References
  • Show All

Further Information

Bioactivity:
TAPI-1 is an ADAM17/TACE inhibitor, which blocks shedding of cytokine receptors.
CAS:
T4122
Formula:
C28H38F3N5O7
Molecular Weight:
613.62
Pathway:
Proteases/Proteasome
Purity:
0.9806
SMILES:
OC(=O)C(F)(F)F.CC(C)CC(CC(=O)NO)C(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)N[C@@H](C)C(=O)NCCN
Target:
MMP

References

M?llberg J, et al. J Immunol. 1995, 155(11), 5198-5205 Oikawa H, et al. Life Sci. 2014, 97(2), 137-144. Slack BE, et al. Biochem J. 2001, 357(Pt 3), 787-794.