TargetMol

Dimethindene

Product Code:
 
TAR-T31488
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T31488-1mg1mg£227.00
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TAR-T31488-2mg2mg£306.00
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TAR-T31488-5mg5mg£431.00
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TAR-T31488-10mg10mg£600.00
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TAR-T31488-25mg25mg£863.00
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TAR-T31488-50mg50mg£1,187.00
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TAR-T31488-100mg100mg£1,581.00
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This product comes from: United States.
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Further Information

Bioactivity:
Dimethindene is a selective antagonist of H1 receptor and blocks K+ current. Dimethindene exhibits antihistamine and anticholinergic effects.
CAS:
5636-83-9
Formula:
C20H24N2
Molecular Weight:
292.42
Pathway:
GPCR/G Protein; Membrane transporter/Ion channel; Immunology/Inflammation; Metabolism; Neuroscience
Purity:
0.9944
SMILES:
N=1C=CC=CC1C(C=2C=3C=CC=CC3CC2CCN(C)C)C
Target:
Potassium Channel; Endogenous Metabolite; AChR; Histamine Receptor

References

1. Sakuta H. Inhibition by histamine H1 receptor antagonists of endogenous glibenclamide-sensitive K+ channels in follicle-enclosed Xenopus oocytes. Eur J Pharmacol. 1994 Jan 1;266(1):99-102. 2. Weller K, et, al. Mast cells are required for normal healing of skin wounds in mice. FASEB J. 2006 Nov;20(13):2366-8. 3. Mikus P, et al. Determination of dimethindene enantiomers in pharmaceuticals by capillary electrophoresis with carboxyethyl-beta-cyclodextrin. Pharmazie. 2007 Jan;62(1):31-3. 4. Schaffler K, et al. Dimethindene maleate in the treatment of sunburn. A double-blind, placebo-controlled pilot study. Arzneimittelforschung. 1999 Apr;49(4):374-9.