TargetMol

Takeda103A

Product Code:
 
TAR-T24850
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T24850-1mg1mg£193.00
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TAR-T24850-5mg5mg£309.00
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TAR-T24850-1mL1 mL * 10 mM (in DMSO)£382.00
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TAR-T24850-10mg10mg£433.00
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TAR-T24850-25mg25mg£667.00
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TAR-T24850-50mg50mg£914.00
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Quantity:
TAR-T24850-100mg100mg£1,187.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
Takeda103A is the GRK2-dependent bovine tubulin oxidation effective inhibitor.
CAS:
865609-72-9
Formula:
C24H23F2N7O
Molecular Weight:
463.493
Pathway:
GPCR/G Protein
Purity:
0.9801
SMILES:
CCCn1c(CNc2cccc(c2)C(=O)NCc2c(F)cccc2F)nnc1-c1ccncn1
Target:
GRK

References

1. Waldschmidt HV, Homan KT, Cruz-Rodr?guez O, et al. Structure-Based Design, Synthesis, and Biological Evaluation of Highly Selective and Potent G Protein-Coupled Receptor Kinase 2 Inhibitors. J Med Chem. 2016 Apr 28;59(8):3793-807. doi: 10.1021/acs.jmedchem.5b02000. Epub 2016 Apr 13. PubMed PMID: 27050625.