TargetMol

Fananserin

Product Code:
 
TAR-T15270
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T15270-1mg1mg£112.00
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TAR-T15270-5mg5mg£155.00
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TAR-T15270-1mL1 mL * 10 mM (in DMSO)£171.00
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TAR-T15270-10mg10mg£189.00
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TAR-T15270-25mg25mg£264.00
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TAR-T15270-50mg50mg£356.00
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TAR-T15270-100mg100mg£495.00
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TAR-T15270-500mg500mg£1,018.00
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Further Information

Bioactivity:
Fananserin is an effective, selective and oral active antagonist of 5-HT2 (Ki = 0.37 nM for the rat 5-HT2A). Fananserin is an antagonist of human D4 receptor (Ki = 2.93 nM).
CAS:
127625-29-0
Formula:
C23H24FN3O2S
Molecular Weight:
425.52
Pathway:
Neuroscience; GPCR/G Protein
Purity:
0.98
SMILES:
Fc1ccc(cc1)N1CCN(CCCN2c3cccc4cccc(c34)S2(=O)=O)CC1
Target:
Dopamine Receptor; 5-HT Receptor

References

1. Malgouris C, et al. Autoradiographic studies of RP 62203, a potent 5-HT2 receptor antagonist. In vitro and ex vivo selectivity profile. Eur J Pharmacol. 1993 Mar 16;233(1):29-35. 2. Stutzmann JM, et al. RP 62203, a 5-hydroxytryptamine2 antagonist, enhances deep NREM sleep in rats. Sleep. 1992 Apr;15(2):119-24. 3. Heuillet E, et al. The naphtosultam derivative RP 62203 (fananserin) has high affinity for the dopamine D4 receptor. Eur J Pharmacol. 1996 Oct 24;314(1-2):229-33.