TargetMol

Esaxerenone

Product Code:
 
TAR-T15246
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T15246-1mg1mg£122.00
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TAR-T15246-5mg5mg£189.00
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TAR-T15246-1mL1 mL * 10 mM (in DMSO)£201.00
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TAR-T15246-10mg10mg£262.00
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TAR-T15246-25mg25mg£442.00
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TAR-T15246-50mg50mg£663.00
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TAR-T15246-100mg100mg£1,002.00
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TAR-T15246-500mg500mg£1,934.00
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This product comes from: United States.
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Further Information

Bioactivity:
Esaxerenone is a highly potent and selective non-steroidal antagonist of the mineralocorticoid receptor.
CAS:
1632006-28-0
Formula:
C22H21F3N2O4S
Molecular Weight:
466.48
Pathway:
Endocrinology/Hormones
Purity:
0.9968
SMILES:
Cc1c(cn(CCO)c1-c1ccccc1C(F)(F)F)C(=O)Nc1ccc(cc1)S(C)(=O)=O
Target:
Glucocorticoid Receptor

References

1. Yamada M, et al. Pharmacokinetics, distribution, and disposition of esaxerenone, a novel, highly potent and selective non-steroidal mineralocorticoid receptor antagonist, in rats and monkeys. Xenobiotica. 2017 Dec;47(12):1090-1103.