TargetMol

LIT-001

Product Code:
 
TAR-T11857
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T11857-1mg1mg£122.00
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TAR-T11857-5mg5mg£195.00
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TAR-T11857-1mL1 mL * 10 mM (in DMSO)£250.00
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TAR-T11857-10mg10mg£301.00
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TAR-T11857-25mg25mg£436.00
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TAR-T11857-50mg50mg£610.00
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TAR-T11857-100mg100mg£838.00
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TAR-T11857-500mg500mg£1,613.00
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Further Information

Bioactivity:
LIT-001 improves social interaction in a mouse model of autism.It is the first nonpeptide oxytocin receptor agonist with EC50 of 55 nM and Ki of 226 nM.
CAS:
2245072-21-1
Formula:
C30H34F3N7O4S
Molecular Weight:
645.7
Pathway:
Endocrinology/Hormones; GPCR/G Protein
Purity:
0.9825
SMILES:
OC(=O)C(F)(F)F.CN(C)C(=S)[C@@H]1CCCN1C(=O)NCc1ccc(cc1C)C(=O)N1Cc2cnn(C)c2Nc2ccccc12
Target:
Oxytocin Receptor

References

1. Frantz MC, et al. LIT-001, the First Nonpeptide Oxytocin Receptor Agonist that Improves Social Interaction in a Mouse Model of Autism. J Med Chem. 2018 Oct 11;61(19):8670-8692.