TargetMol

IPR-803

Product Code:
 
TAR-T11666
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T11666-1mg1mg£138.00
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TAR-T11666-5mg5mg£229.00
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TAR-T11666-1mL1 mL * 10 mM (in DMSO)£252.00
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TAR-T11666-10mg10mg£334.00
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TAR-T11666-25mg25mg£519.00
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TAR-T11666-50mg50mg£703.00
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Further Information

Bioactivity:
IPR-803 is an effective inhibitor of the uPAR?uPA protein-protein interaction (PPI) with anti-tumor activity. IPR-803 binds directly to uPAR with a Ki of 0.2 μM.
CAS:
892243-35-5
Formula:
C27H23N3O4
Molecular Weight:
453.498
Pathway:
Metabolism; Cell Cycle/Checkpoint
Purity:
0.98
SMILES:
OC(=O)c1cccc(Nc2cc(N3CCCCCC3)c3noc4-c5ccccc5C(=O)c2c34)c1
Target:
Serine/threonin kinase

References

1. Mani T, et al. Small-molecule inhibition of the uPAR?uPA interaction: synthesis, biochemical, cellular, in vivo pharmacokinetics and efficacy studies in breast cancer metastasis. Bioorg Med Chem. 2013 Apr 1;21(7):2145-55.