TargetMol

Eplivanserin

Product Code:
 
TAR-T11217
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T11217-1mg1mg£227.00
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TAR-T11217-5mg5mg£422.00
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TAR-T11217-1mL1 mL * 10 mM (in DMSO)£426.00
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TAR-T11217-10mg10mg£589.00
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TAR-T11217-25mg25mg£863.00
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TAR-T11217-50mg50mg£1,179.00
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This product comes from: United States.
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Further Information

Bioactivity:
Eplivanserin is an effective and selective antagonist of 5-HT2A receptor with a Kd of 1.14 nM and an IC50 value of 5.8 nM in rat cortical membrane.
CAS:
130579-75-8
Formula:
C19H21FN2O2
Molecular Weight:
328.387
Pathway:
GPCR/G Protein; Neuroscience
Purity:
0.98
SMILES:
CN(C)CCON=C(C=Cc1ccc(O)cc1)/c1ccccc1F
Target:
5-HT Receptor

References

1. Malgorzata Filip, et al. Contribution of serotonin (5-hydroxytryptamine; 5-HT) 5-HT2 receptor subtypes to the hyperlocomotor effects of cocaine: acute and chronic pharmacological analyses. J Pharmacol Exp Ther. 2004 Sep;310(3):1246-54. 2. Rinaldi-Carmona M, et al. Biochemical and pharmacological properties of SR 46349B, a new potent and selective 5-hydroxytryptamine2 receptor antagonist. J Pharmacol Exp Ther. 1992 Aug;262(2):759-68.