TargetMol

Ecopladib

Product Code:
 
TAR-T11149
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T11149-1mg1mg£1,420.00
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TAR-T11149-5mg5mg£2,769.00
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TAR-T11149-10mg10mg£3,709.00
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TAR-T11149-1mL1 mL * 10 mM (in DMSO)£4,801.00
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TAR-T11149-25mg25mg£5,492.00
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TAR-T11149-50mg50mg£7,243.00
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TAR-T11149-100mg100mg£9,950.00
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Further Information

Bioactivity:
Ecopladib with IC50s of 0.15 μM and 0.11 μM in the GLU micelle and rat whole blood assays, respectively.Ecopladib is a sub-micromolar inhibitor of cytosolic phospholipase A2α (cPLA2α).
CAS:
381683-92-7
Formula:
C39H33Cl3N2O5S
Molecular Weight:
748.11
Pathway:
Metabolism
Purity:
0.98
SMILES:
OC(=O)c1ccc(OCCc2c(CCNS(=O)(=O)Cc3ccc(Cl)c(Cl)c3)n(C(c3ccccc3)c3ccccc3)c3ccc(Cl)cc23)cc1
Target:
Phospholipase

References

1. Lee KL, et al. Discovery of Ecopladib, an indole inhibitor of cytosolic phospholipase A2alpha. J Med Chem. 2007 Mar 22;50(6):1380-400. Epub 2007 Feb 17.