TargetMol

3-Bromocytisine

Product Code:
 
TAR-T10108
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T10108-1mg1mg£148.00
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Quantity:
TAR-T10108-1mL1 mL * 10 mM (in DMSO)£246.00
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TAR-T10108-5mg5mg£262.00
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TAR-T10108-10mg10mg£332.00
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TAR-T10108-25mg25mg£511.00
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TAR-T10108-50mg50mg£703.00
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Quantity:
TAR-T10108-100mg100mg£938.00
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This product comes from: United States.
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Further Information

Bioactivity:
3-Bromocytisine is an effective agonist of nAChR (IC50s: 0.28, 0.30 and 31.6 nM for hα4β4, hα4β2, and hα7).
CAS:
207390-14-5
Formula:
C11H13BrN2O
Molecular Weight:
269.14
Pathway:
Neuroscience
Purity:
0.9814
SMILES:
O=C1N2C([C@@]3(C[C@](C2)(CNC3)[H])[H])=CC=C1Br
Target:
AChR

References

1. Houlihan LM, et al. Activity of cytisine and its brominated isosteres on recombinant human alpha7, alpha4beta2 and alpha4beta4 nicotinic acetylcholine receptors. J Neurochem. 2001 Sep;78(5):1029-43. 2. Moroni M, et al. alpha4beta2 nicotinic receptors with high and low acetylcholine sensitivity: pharmacology, stoichiometry, and sensitivity to long-term exposure to nicotine. Mol Pharmacol. 2006 Aug;70(2):755-68.